1G244

• Target :

  Apoptosis|||Proteasome

• Related Pathways :

  Ubiquitination|||Proteases/Proteasome|||Apoptosis

• Purity :

  0.9914

• Bioactivity :

  1G244 is an inhibitor of DPP8/9 with antiatherosclerotic and antimyeloma properties. 1G244 had the IC50 values of 14 and 53 nM against DPP8 and DPP9, and The Ki values for 1G244 were 0.9 and 4.2 nM for DPP8 and DPP9

• Smiles :

  N[C@@H](CC(=O)N1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)N1Cc2ccccc2C1

• Molecular Formula :

  C29H30F2N4O2

• Molecular Weight :

  504.57

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  847928-32-9