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VTP50469

CAT: 0931-T13336-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T13336-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2169916-18-9
Target
Histone Methyltransferase, Epigenetic Reader Domain, Apoptosis
Related Pathways
Apoptosis, Chromatin/Epigenetic
Purity
0.9955
Bioactivity
VTP50469 is a highly selective and orally active small molecule inhibitor of the Menin-MLL protein-protein interaction with potent anti-leukemic activity with a Ki of 104 pM.
Smiles
CC(C)N(C(C)C)C(=O)c1cc(F)ccc1Oc1cncnc1N1CC2(C1)CCN(C[C@H]1CC[C@@H](CC1)NS(C)(=O)=O)CC2
Molecular Formula
C32H47FN6O4S
Molecular Weight
630.82
Shipping Conditions
Ice Packs
Storage Temperature
-20°C