TPA-023B

• Target:

  Others|||GABA Receptor

• Related Pathways:

  Neuroscience|||Membrane transporter/Ion channel|||Others

• Bioactivity:

  TPA-023B is an orally active and high-affinity agonist of the GABAA receptor ?2/?3 subtype (Kis: 0.73 nM/2 nM) partial and an antagonist ?1 subtype (Ki: 1.8 nM), has non-sedating anxiolytic-like properties.

• Smiles:

  CC(C)(O)c1cnn2c(cnc2n1)-c1ccc(F)c(c1)-c1c(F)cccc1C#N

• Molecular Formula:

  C21H15F2N5O

• Molecular Weight:

  391.37

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  425377-76-0