TPA-023B

CAT: 0931-T13192-01Size: 25 mgDry Ice: NoHazardous: No
CAT#: T13192-01Size: 25 mg
Selected
AVAILABILITY
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
425377-76-0
Target
Others|||GABA Receptor
Related Pathways
Neuroscience|||Membrane transporter/Ion channel|||Others
Bioactivity
TPA-023B is an orally active and high-affinity agonist of the GABAA receptor ?2/?3 subtype (Kis: 0.73 nM/2 nM) partial and an antagonist ?1 subtype (Ki: 1.8 nM), has non-sedating anxiolytic-like properties.
Smiles
CC(C)(O)c1cnn2c(cnc2n1)-c1ccc(F)c(c1)-c1c(F)cccc1C#N
Molecular Formula
C21H15F2N5O
Molecular Weight
391.37
Shipping Conditions
Cool pack
Storage Temperature
-20°C