J-2156

• Target :

  Others|||Somatostatin

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. J-2156 is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively.

• Smiles :

  S(N[C@H](C(N[C@@H](CC1=CC=CC=C1)C(N)=O)=O)CCN)(=O)(=O)C=2C3=C(C(C)=CC2)C=CC=C3

• Molecular Formula :

  C24H28N4O4S

• Molecular Weight :

  468.57

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  848647-56-3