Products for Research Use Only

GSK3368715

CAT: 0931-T11500-01Size: 100 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T11500-01Size:100 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1629013-22-4
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8) ) . It has strong anti-cancer activity.
Smiles
C(OCC)C1(COCC)CCC(CC1)C=2C(CN(CCNC)C)=CNN2
Molecular Formula
C20H38N4O2
Molecular Weight
366.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C