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GCN2-IN-6

CAT: 0931-T11374-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T11374-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2183470-09-7
Target
PERK
Related Pathways
Apoptosis
Purity
0.98
Bioactivity
GCN2-IN-6 is a potent and orally available GCN2 inhibitor confirmed by in-house enzymatic (IC50: 1.8 nM) and cellular assays (IC50: 9.3 nM) . GCN2-IN-6 is also an eIF2α kinase PERK inhibitor with IC50s of 0.26 nM in enzymatic assay and 230 nM in cells respectively.
Smiles
Nc1ncc(cn1)C#Cc1c(F)ccc(NS(=O)(=O)c2cc(Cl)cc(CO)c2Cl)c1F
Molecular Formula
C19H12Cl2F2N4O3S
Molecular Weight
485.29
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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