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ERRα antagonist-1

CAT: 0931-T11230-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T11230-01Size:2 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1072145-33-5
Target
Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Related Pathways
Endocrinology/Hormones
Purity
>99.99%
Bioactivity
ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα) . It effectively prevents the interaction of ERRα with both Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, displaying IC50 values of 170 nM and 180 nM, respectively. Notably, ERRα antagonist-1 does not interfere with the interactions involving ERRβ or ERRγ and the PGC-1α and PGC-1β coactivators. Furthermore, it does not affect the interaction between either ERα or ERβ and PGC-1α or SRC-1.
Smiles
C1CN=C(S1)N1CCS\C1=N/C1c2ccccc2C=Cc2ccccc12
Molecular Formula
C21H19N3S2
Molecular Weight
377.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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Alternative Products

CatalogName
A9977-25ERRα antagonist-1
GTR19186597-01ERRα antagonist-2
HY-145848-01ERRγ agonist-1
sc-393969ERRγ (D-1)
sc-376449ERRβ/γ (E-1)
M23437-01PROTAC ERRα ligand 1
HY-128838-01PROTAC ERRα Degrader-1
sc-376449 PEERRβ/γ (E-1) PE
sc-393969 XERRγ (D-1) X
sc-376449 FITCERRβ/γ (E-1) FITC

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