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ERRα antagonist-1

CAT: 0931-T11230-01Size: 2 mgDry Ice: NoHazardous: No
CAT#:0931-T11230-01Size:2 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1072145-33-5
Target
Estrogen Receptor/ERR|||Estrogen/progestogen Receptor
Related Pathways
Endocrinology/Hormones
Purity
>99.99%
Bioactivity
ERR? antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor ? (ERR?) . It effectively prevents the interaction of ERR? with both Proliferator-activated Receptor ? Coactivator-1? (PGC-1?) and PGC-1?, displaying IC50 values of 170 nM and 180 nM, respectively. Notably, ERR? antagonist-1 does not interfere with the interactions involving ERR? or ERR? and the PGC-1? and PGC-1? coactivators. Furthermore, it does not affect the interaction between either ER? or ER? and PGC-1? or SRC-1.
Smiles
C1CN=C(S1)N1CCS\C1=N/C1c2ccccc2C=Cc2ccccc12
Molecular Formula
C21H19N3S2
Molecular Weight
377.53
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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