BI-9321

• Target:

  Others|||Histone Methyltransferase

• Related Pathways:

  Others|||Chromatin/Epigenetic

• Bioactivity:

  BI-9321 is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3) -PWWP1 domain antagonist (Kd: 166 nM) . BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2.

• Smiles:

  CN1C(=C(N=C1)C2=C(C)C=C(CN)C=C2C)C=3C4=C(C=C(F)C=C4)N=CC3

• Molecular Formula:

  C22H21FN4

• Molecular Weight:

  360.43

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2387510-86-1