BI-9321
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


BI-9321
Target :
Others|||Histone MethyltransferaseRelated Pathways :
Others|||Chromatin/EpigeneticBioactivity :
BI-9321 is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3) -PWWP1 domain antagonist (Kd: 166 nM) . BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2.Smiles :
CN1C(=C(N=C1)C2=C(C)C=C(CN)C=C2C)C=3C4=C(C=C(F)C=C4)N=CC3Molecular Formula :
C22H21FN4Molecular Weight :
360.43Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
2387510-86-1

