GF109203X ,PKC kinase inhibitor
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Catalog numberSIH-447-10MG
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PricePlease ask
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Size10 mg
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Research Area sCell Signaling , Cancer , Apoptosis , Cancer Growth Inhibitors , Tyrosine Kinase Inhibitors
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CategorySmall Molecules
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Product TypeInhibitor
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CAS No133052-90-1
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MolecularFormulaC25H24N4O2
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Molecular Weight412.5
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Purity≥98% (TLC)
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SolubilitySoluble in dimethyl formamide or DMSO (10 mg/ml, warm to 40°C and vortex well)
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AppearanceRed solid
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Storage Temperature-20°C
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Shipping TemperatureShipped Ambient
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DescriptionTissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
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Gene target
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Gene symbolPRKCH, PRKD1, PRRT2, PRKDC
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Short nameGF109203X ,PKC kinase inhibitor
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Alternative nameGF109203X ,PKC phosphorylation catalyst suppressor
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Gene info
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Identity
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Gene
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Long gene nameprotein kinase C eta
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Synonyms gene
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Synonyms gene name
- protein kinase C, eta
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Synonyms
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GenBank acession
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Locus
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Discovery year1992-06-26
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
- C2 domain containing protein kinases
- AGC family kinases
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VEGA ID
Gene info
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Identity
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Gene
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Long gene nameprotein kinase D1
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Synonyms gene
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Synonyms gene name
- protein kinase C, mu
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Synonyms
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Locus
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Discovery year1994-05-16
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
- Pleckstrin homology domain containing
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VEGA ID
Gene info
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Identity
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Gene
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Long gene nameproline rich transmembrane protein 2
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Synonyms gene
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Synonyms gene name
- infantile convulsions and paroxysmal choreoathetosis
- dystonia 10
- proline-rich transmembrane protein 2
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Synonyms
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Synonyms name
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GenBank acession
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Locus
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Discovery year2005-11-25
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
- interferon induced transmembrane protein domain containing
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VEGA ID
Gene info
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Identity
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Gene
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Long gene nameprotein kinase, DNA-activated, catalytic subunit
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Synonyms gene
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Synonyms gene name
- protein kinase, DNA-activated, catalytic polypeptide
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Synonyms
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Synonyms name
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Locus
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Discovery year1993-11-09
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Entrez gene record
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Pubmed identfication
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RefSeq identity
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Classification
- Armadillo like helical domain containing
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VEGA ID
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Locus Specific Databases