6BIO,PDK1 kinase inhibitor
-
Catalog numberSIH-422-25MG
-
PricePlease ask
-
Size25 mg
-
-
Research Area sCell Signaling
-
CategorySmall Molecules
-
Product TypeInhibitor
-
CAS No667463-62-9
-
MolecularFormulaC16H10BrN3O2
-
Molecular Weight356.2
-
Purity≥98% (HPLC)
-
SolubilitySoluble to 10 mM in DMSO and to 10 mM in ethanol
-
AppearanceDark red solid
-
Storage Temperature-20°C
-
Shipping TemperatureShipped Ambient
-
DescriptionTissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
-
Gene target
-
Gene symbolPDK1, PDPK1
-
Short name6BIO PDK1 kinase inhibitor
-
Alternative name6BIO,PDK1 phosphorylation catalyst suppressor
-
Gene info
-
Identity
-
Gene
-
Long gene namepyruvate dehydrogenase kinase 1
-
Synonyms gene name
- pyruvate dehydrogenase kinase, isoenzyme 1
- pyruvate dehydrogenase kinase, isozyme 1
-
GenBank acession
-
Locus
-
Discovery year1996-08-14
-
Entrez gene record
-
Pubmed identfication
-
RefSeq identity
-
VEGA ID
Gene info
-
Identity
-
Gene
-
Long gene name3-phosphoinositide dependent protein kinase 1
-
Synonyms
-
Synonyms name
-
GenBank acession
-
Locus
-
Discovery year1998-03-23
-
Entrez gene record
-
Pubmed identfication
-
Classification
- AGC family kinases
-
VEGA ID