K252a
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Catalog number2013-1000
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PricePlease ask
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Size1 mg
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Alternative_nameSF 2370
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DescriptionAn analog of Staurosporine (Cat. No. 1048) that acts as a non-selective protein kinase inhibitor. Iinhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), and PKG (Ki = 20 nM). Potently inhibits CaMK (Ki = 1.8 nM), competitively with ATP and noncompetitively with the substrate.
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CAS Number99533-80-9
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Structure AvailableYes
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Salt FormNo
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Molecular FormulaC₂₇H₂₁N₃O₅
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Molecular Weight467.47
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO (100 mg/ml)
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HandlingProtect from air and light
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Tag LineA selective protein kinase inhibitor
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Storage Condition-20°C
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Shipping Conditiongel pack
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Shelf Life24months
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MDL NumberMFCD00161522
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PubChem CID127357
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SMILESCC12C(CC(O1)N3C4=CC=CC=C4C5=C6C(=C7C8=CC=CC=C8N2C7=C53)CNC6=O)(C(=O)OC)O
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InChi KeyKOZFSFOOLUUIGY-UHOLRESSSA-N
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MSDS AvailableYes
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Gene target
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Short nameK252a
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Alternative nameK252a
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