K252a

  • Catalog number
    2013-1000
  • Price
    Please ask
  • Size
    1 mg
  • Alternative_name
    SF 2370
  • Description
    An analog of Staurosporine (Cat. No. 1048) that acts as a non-selective protein kinase inhibitor. Iinhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), and PKG (Ki = 20 nM). Potently inhibits CaMK (Ki = 1.8 nM), competitively with ATP and noncompetitively with the substrate.
  • CAS Number
    99533-80-9
  • Structure Available
    Yes
  • Salt Form
    No
  • Molecular Formula
    C₂₇H₂₁N₃O₅
  • Molecular Weight
    467.47
  • Cell Permeable
    Yes
  • Purity
    ≥98% by HPLC
  • Solubilities
    DMSO (100 mg/ml)
  • Handling
    Protect from air and light
  • Tag Line
    A selective protein kinase inhibitor
  • Storage Condition
    -20°C
  • Shipping Condition
    gel pack
  • Shelf Life
    24months
  • MDL Number
    MFCD00161522
  • PubChem CID
    127357
  • SMILES
    CC12C(CC(O1)N3C4=CC=CC=C4C5=C6C(=C7C8=CC=CC=C8N2C7=C53)CNC6=O)(C(=O)OC)O
  • InChi Key
    KOZFSFOOLUUIGY-UHOLRESSSA-N
  • MSDS Available
    Yes
  • Gene target
    K252a  
  • Short name
    K252a
  • Alternative name
    K252a
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