CB-839

• Catalog number
  B1179-5
• Price
  Please ask
• Size
  5 mg

• Alternative_name
  2-(pyridin-2-yl)-N-(5-(4-(6-(2-(3-(trifluoromethoxy)phenyl)acetamido)pyridazin-3-yl)butyl)-1,3,4-thiadiazol-2-yl)acetamide
• Description
  CB-839 is a potent, selective, and orally bioavailable inhibitor of both splice variants of glutaminase (KGA and GAC); inhibits recombinant GAC with an IC₅₀ of
• CAS Number
  1439399-58-2
• Structure Available
  Yes
• Molecular Formula
  C₂₆H₂₄F₃N₇O₃S
• Molecular Weight
  571.57
• Cell Permeable
  Yes
• Purity
  ≥97% by HPLC
• Solubilities
  DMSO
• Handling
  Protect from air and light
• Tag Line
  A potent glutaminase inhibitor
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• PubChem CID
  71577426
• PubChem CID Link
• SMILES
  C1=CC=NC(=C1)CC(=O)NC2=NN=C(S2)CCCCC3=NN=C(C=C3)NC(=O)CC4=CC(=CC=C4)OC(F)(F)F
• InChi
  InChI=1S/C26H24F3N7O3S/c27-26(28,29)39-20-9-5-6-17(14-20)15-22(37)31-21-12-11-18(33-34-21)7-1-2-10-24-35-36-25(40-24)32-23(38)16-19-8-3-4-13-30-19/h3-6,8-9,11-14H,1-2,7,10,15-16H2,(H,31,34,37)(H,32,36,38)
• InChi Key
  PRAAPINBUWJLGA-UHFFFAOYSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  CB-839  
• Gene symbol
  CNR1
• Short name
  CB-839
• Alternative name
  CB-839

Gene info

• Identity
  HGNC:2159
• Gene
  CNR1
• Long gene name
  cannabinoid receptor 1
• Synonyms gene
  • CNR
• Synonyms gene name
  • cannabinoid receptor 1 (brain)
• Synonyms
  • CB1K5
  • CB-R
  • CB1
  • CANN6
  • CB1A
• GenBank acession
  • AF107262
• Locus
  6q15
• Discovery year
  1991-05-15
• Entrez gene record
  1268
• Classification
  • Cannabinoid receptors
• VEGA ID
  OTTHUMG00000015184

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