PHA 665752,MET kinase inhibitor
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Catalog numberSIH-421-25MG
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PricePlease ask
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Size25 mg
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Research Area sCell Signaling , Cancer , Apoptosis , Cancer Growth Inhibitors , Tyrosine Kinase Inhibitors
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CategorySmall Molecules
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Product TypeInhibitor
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CAS No477575-56-7
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MolecularFormulaC32H34Cl2N4O4S
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Molecular Weight641.61
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Purity>98
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SolubilitySoluble to 100 mM in DMSO.
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AppearanceYellow solid
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Storage Temperature-20°C
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Shipping TemperatureShipped Ambient
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DescriptionTissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
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Gene target
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Gene symbolSLTM, MET, TRM-CAT4-3, TRM-CAT5-1, TRM-CAT3-2, TRM-CAT7-1, TRM-CAT5-2, TRM-CAT2-1, TRM-CAT3-1, TRM-CAT4-2
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Short namePHA 665752 MET kinase inhibitor
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Alternative namePHA 665752,MET phosphorylation catalyst suppressor
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Gene info
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Identity
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Gene
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Long gene nameSAFB like transcription modulator
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Synonyms
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GenBank acession
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Locus
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Discovery year2005-11-08
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Entrez gene record
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RefSeq identity
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Classification
- RNA binding motif containing
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VEGA ID
Gene info
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Identity
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Gene
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Long gene nameMET proto-oncogene, receptor tyrosine kinase
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Synonyms gene name
- met proto-oncogene
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Synonyms
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Synonyms name
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GenBank acession
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Locus
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Discovery year1986-01-01
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Pubmed identfication
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Classification
- Receptor tyrosine kinases
- IPT domain containing
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VEGA ID
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Locus Specific Databases
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 4-3
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 20 (anticodon CAU)
- transfer RNA-Met (CAT) 4-3
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 5-1
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 16 (anticodon CAU)
- transfer RNA-Met (CAT) 5-1
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 3-2
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 8 (anticodon CAU)
- transfer RNA-Met (CAT) 3-2
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 7-1
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 5 (anticodon CAU)
- transfer RNA-Met (CAT) 7-1
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 5-2
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Synonyms
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Locus
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Discovery year2019-12-06
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 2-1
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 9 (anticodon CAU)
- transfer RNA-Met (CAT) 2-1
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 3-1
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 12 (anticodon CAU)
- transfer RNA-Met (CAT) 3-1
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs
Gene info
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Identity
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Gene
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Long gene nametRNA-Met (anticodon CAT) 4-2
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Synonyms gene
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Synonyms gene name
- transfer RNA methionine 19 (anticodon CAU)
- transfer RNA-Met (CAT) 4-2
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Synonyms
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GenBank acession
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Locus
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Discovery year2008-08-29
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Entrez gene record
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Classification
- Cytoplasmic transfer RNAs