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GA001

CAT: 0804-HY-164479Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-164479Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GA001 is a potent G9a antagonist, with an IC50 of 1.32 μM. GA001 induces autophagy and apoptosis that can be used for the breast cancer[1].
CAS Number
2097880-27-6
UNSPSC
12352005
Target
Apoptosis; Autophagy; Histone Methyltransferase
Type
Reference compound
Related Pathways
Apoptosis; Autophagy; Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ga001.html
Smiles
O=C(C1=CC(Br)=CC=C1)NC2=CC=C3C(N=C(N3CCCC4=CC=CC=C4)C5=CC=CC=C5)=C2
Molecular Formula
C29H24BrN3O
Molecular Weight
510.42
References & Citations
[1]Zhang J, et al. Synthesis and biological evaluation of benzimidazole derivatives as the G9a Histone Methyltransferase inhibitors that induce autophagy and apoptosis of breast cancer cells. Bioorg Chem. 2017 Jun;72:168-181.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Alternative Products

CatalogName
GTR19239030-01GA001

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