CYB210010

CAT: 0804-HY-162423Size: 1 EachDry Ice: NoHazardous: No

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CAT#:0804-HY-162423Size:1 Each

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Description

CYB210010 is an orally bioavailable, long-acting serotonin 5-HT2 receptor agonist that selectively targets 5-HT2A and 5-HT2C receptors (EC50: 4.1 n, 7.3 nM) . CYB210010 can enter the central nervous system, cause a head twitch response (HTR), and is not prone to behavioral tolerance during chronic administration[1].

CAS Number

2762568-47-6

UNSPSC

12352005

Target

5-HT Receptor; Androgen Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling; Vitamin D Related/Nuclear Receptor

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/cyb210010.html

Solubility

10 mM in DMSO

Smiles

COC1=C(CCN)C=C(OC)C(SC(F)(F)F)=C1.Cl

Molecular Formula

C11H15ClF3NO2S

Molecular Weight

317.76

References & Citations

[1]Varty GB, et al. Synthesis and Structure-Activity Relationships of 2,5-Dimethoxy-4-Substituted Phenethylamines and the Discovery of CYB210010: A Potent, Orally Bioavailable and Long-Acting Serotonin 5-HT2 Receptor Agonist. J Med Chem. 2024 Apr 25;67 (8) :6144-6188.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

5-HT2 Receptor; mLAG-3; MUC2; MUC3; α-1 microglobulin

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Catalog	Name
GTR19235530-01	CYB210010

CYB210010

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