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CLP-3094

CAT: 0804-HY-141487-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-141487-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CLP-3094 is a potent BF3 (binding function 3) -directed inhibitor of the androgen receptor (AR) . CLP-3094 inhibits AR transcriptional activity (IC50=4 μM) [1]. CLP-3094 is a selective, potent GPR142 antagonist[2].
CAS Number
312749-73-8
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Androgen Receptor
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Metabolic Disease; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/clp-3094.html
Purity
99.92
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
ClC1=CC=C(OCCSC2=NC3=CC=CC=C3N2)C=C1
Molecular Formula
C15H13ClN2OS
Molecular Weight
304.79
Precautions
H302, H315, H319, H335
References & Citations
[1]Munuganti RS, et al. Targeting the binding function 3 (BF3) site of the androgen receptor through virtual screening. 2. development of 2- ((2-phenoxyethyl) thio) -1H-benzimidazole derivatives. J Med Chem. 2013;56 (3) :1136-1148.|[2]Murakoshi M, et al. Discovery and pharmacological effects of a novel GPR142 antagonist. J Recept Signal Transduct Res. 2017;37 (3) :290-296.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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