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Balovaptan

CAT: 0804-HY-109024-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-109024-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Balovaptan (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism.
CAS Number
1228088-30-9
Product Name Alternative
RG7314
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Vasopressin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease; Endocrinology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/Balovaptan.html
Purity
99.89
Solubility
DMSO : 50 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
CN1CC2=NN=C([C@H]3CC[C@H](OC4=NC=CC=C4)CC3)[N@]2[C@]5=CC=C(Cl)C=C5C1
Molecular Formula
C22H24ClN5O
Molecular Weight
409.91
Precautions
H302, H315, H319, H335
References & Citations
[1]Ratni H, et al. Discovery of highly selective brain-penetrant vasopressin 1a antagonists for the potential treatment of autism via a chemogenomic and scaffold hopping approach. J Med Chem. 2015 Mar 12;58 (5) :2275-89.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 3
Isoform
V1a Receptor

Alternative Products

CatalogName
BA5834-5.1Balovaptan
A19373-100Balovaptan 100mg
A19373-25Balovaptan 25mg
A19373-10Balovaptan 10mg
A19373-5Balovaptan 5mg
A19373-50Balovaptan 50mg
A19373-1Balovaptan 1mg
A19373-10mM-DBalovaptan 10mM * 1mL in DMSO

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