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ASP7663

CAT: 0026-B2976-25Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0026-B2976-25Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
ASP7663 is a selective transient receptor potential ankyrin 1 (TRPA1) activator. It activates human, rat and mouse TRPA1 receptors with EC₅₀ values of 510 nM, 540 nM and 500 nM, respectively. It releases 5-HT from QGP-1 cells. It enhances colonic motility and exerts anti-constipation, analgesic effects against abdominal pain in vivo.
Shipping Conditions
Gel Pack
Storage Conditions
-20ºC
Shelf Life
36months

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