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Thiamet G

CAT: 0026-B2959-5Size: 5 mgDry Ice: NoHazardous: No
CAT#:0026-B2959-5Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Thiamet G is a potent and selective inhibitor of O-GlcNAcase with a Ki value of 21 nM. It increases cellular O-GlcNAc-modified protein levels with an EC₅₀ of 30 nM and blocks phosphorylation of tau protein both in cultured PC-12 cells and in rats (200 mg/kg/day). It is the first highly potent O-GlcNAcase inhibitor known to be orally bioavailable and can effectively cross the blood brain barrier. It may potentially block pathological hyperphosphorylation of tau in Alzheimer's disease.
Shipping Conditions
RT
Storage Conditions
-20ºC
Shelf Life
36 months

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