(±) -Tazifylline

• Description :

  (±) -Tazifylline is a potent, selective and long-acting histamine H1 receptor antagonist.

• UNSPSC :

  12352005

• Target :

  Histamine Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

• Applications :

  Metabolism-protein/nucleotide metabolism

• Field of Research :

  Neurological Disease; Endocrinology

• Assay Protocol :

  https://www.medchemexpress.com/((plusmn))-Tazifylline.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C(N1C)N(C)C2=C(N(CC(O)CN3CCN(CCCSC4=CC=CC=C4)CC3)C=N2)C1=O

• Molecular Formula :

  C23H32N6O3S

• Molecular Weight :

  472.60

• References & Citations :

  [1]Poizot A, et al. Animal pharmacology of the selective histamine H1-receptor antagonist tazifylline. Arzneimittelforschung. 1986 Apr;36 (4) :695-702.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  H1 Receptor

• CAS Number :

  [79712-55-3]