Mianserin

• UNSPSC Description:

  Mianserin is an H1 receptor inverse agonist.

• Target Antigen:

  Histamine Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Neurological Disease; Endocrinology

• Assay Protocol:

  https://www.medchemexpress.com/mianserin.html

• Solubility:

  10 mM in DMSO

• Smiles:

  CN(CC1)CC2N1C3=CC=CC=C3CC4=CC=CC=C24

• Molecular Weight:

  264.36

• References & Citations:

  [1]Olianas MC, et al. The atypical antidepressant mianserin exhibits agonist activity at κ-opioid receptors. Br J Pharmacol. 2012 Nov;167(6):1329-41.|[2]Roeder T. High-affinity antagonists of the locust neuronal octopamine receptor. Eur J Pharmacol. 1990 Nov 27;191(2):221-4.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  Launched

• CAS Number:

  24219-97-4