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Eltoprazine

CAT: 0804-HY-16687Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-16687Size:1 Each
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Description
Eltoprazine (DU 28853) is a 5-HT1A/5-HT1B receptors agonist and a 5-HT2C receptor antagonist. Eltoprazine shows antiaggressive and anxiogenic effects[1][2].
CAS Number
98224-03-4
Product Name Alternative
DU 28853
UNSPSC
12352005
Hazard Statement
H301-H315-H319-H335
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Eltoprazine.html
Purity
95.0
Solubility
DMSO : ≥ 25 mg/mL
Smiles
N1(C2=C3OCCOC3=CC=C2)CCNCC1
Molecular Formula
C12H16N2O2
Molecular Weight
220.27
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362-P403+P233-P405-P501
References & Citations
[1]Sijbesma H, et al. Eltoprazine, a drug which reduces aggressive behaviour, binds selectively to 5-HT1 receptor sites in the rat brain: an autoradiographic study. Eur J Pharmacol. 1990 Feb 20;177 (1-2) :55-66.|[2]Rocha B, et al. Chronic mianserin or eltoprazine treatment in rats: effects on the elevated plus-maze test and on limbic 5-HT2C receptor levels. Eur J Pharmacol. 1994 Sep 1;262 (1-2) :125-31.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 3
Isoform
5-HT1 Receptor;5-HT2 Receptor; mLAG-3; α-1 microglobulin

Alternative Products

CatalogName
T38145-01Eltoprazine
T7498-01Eltoprazine hydrochloride
MBS5758627Eltoprazine dihydrochloride
528830Eltoprazine HCl
A20861-25Eltoprazine 25mg
A20861-10Eltoprazine 10mg
A20861-100Eltoprazine 100mg
A20861-50Eltoprazine 50mg

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