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Siltenzepine

CAT: 0804-HY-101694Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-101694Size:1 Each
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Description
Siltenzepine (AWD 26-06 free base) is an antagonist of mAChR with anti-acid activity, which can be used in peptic ulcers research. Siltenzepine exhibits rapidly but incompletely absorbed characterastic in rats (po) [1][2].
CAS Number
98374-54-0
Product Name Alternative
AWD 26-06 (free base)
UNSPSC
12352005
Target
MAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/Siltenzepine.html
Solubility
10 mM in DMSO
Smiles
O=C1C2=CC=CC=C2N(C(CN(CCO)CCO)=O)C3=CC=C(Cl)C=C3N1
Molecular Formula
C19H20ClN3O4
Molecular Weight
389.83
References & Citations
[1]Pfeifer S, et al. Biotransformation und Pharmakokinetik von AWD 26-06, 8-Chlor-5,10-dihydro-5-[bis (2-hydroxyethyl) aminoacetyl]-11H- dibenzo[d, c][1,4]diazepin-11-on-hydrochlorid an der Ratte [Biotransformation and pharmacokinetics of AWD 26-06, 8-chloro-5,10-dihydro-5-[bis (2-hydroxyethyl) aminoacetyl]-11H-dibenzo[d, c][1,4]diazepin-11-one hydrochloride in the rat]. Pharmazie. 1990 Jul;45 (8) :603-7. German.|[2]Trausch B, et al. The biliary and renal elimination of the new muscarinic-1-antagonist AWD 26-06 in volunteers with T-tube after cholecystectomy. Int J Clin Pharmacol Ther Toxicol. 1992 Nov;30 (11) :508-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Alternative Products

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T12914-01Siltenzepine
A19818-50Siltenzepine 50mg
A19818-25Siltenzepine 25mg
A19818-100Siltenzepine 100mg
A19818-10Siltenzepine 10mg
A19818-5Siltenzepine 5mg
A19818-1Siltenzepine 1mg

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