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Alvameline

CAT: 0804-HY-101586-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-101586-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Alvameline (Lu25-109) is a partial M1 agonist and M2/M3 antagonist.
CAS Number
120241-31-8
Product Name Alternative
Lu 25-109
UNSPSC
12352005
Target
MAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Alvameline.html
Solubility
10 mM in DMSO
Smiles
CN1CCC=C(C2=NN(CC)N=N2)C1
Molecular Formula
C9H15N5
Molecular Weight
193.25
References & Citations
[1]Jensen KG, et al. In vitro metabolism of the M1-muscarinic agonist 5- (2-ethyl-2H-tetrazol-5-yl) -1-methyl-1,2,3,6-tetrahydropyridine by human hepatic cytochromes P-450 determined at pH 7.4 and 8.5. Drug Metab Dispos. 1999 Jan;27 (1) :125-32.|[2]Waldeck K, et al. Actions of the new antimuscarinic compound Alvameline on isolated human and pig detrusor. Neurourol Urodyn. 2002;21 (1) :92-8.|[3]Pike BR, et al. Chronic administration of a partial muscarinic M1 receptor agonist attenuates decreases in forebrain choline acetyltransferase immunoreactivity following experimental brain trauma. Exp Neurol. 1997 Sep;147 (1) :55-65.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
MAChR3

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