Glucagon receptor antagonists-1

• UNSPSC Description:

  Glucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist.

• Target Antigen:

  GCGR

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Metabolism-sugar/lipid metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/glucagon-receptor-antagonists-1.html

• Purity:

  98.65

• Solubility:

  DMSO : 50 mg/mL (ultrasonic)

• Smiles:

  FC1=CC=C(C2=C(/C=C/C)C(C(C)C)=NC(C(C)C)=C2C(C)O)C(OCC3=CC=CC=C3)=C1

• Molecular Weight:

  447.58

• References & Citations:

  [1]Ladouceur, Gaetan H. et al. Integration of optimized substituent patterns to produce highly potent 4-aryl-pyridine glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters (2002), 12(23), 3421-3424.

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  -20°C, 3 years; 4°C, 2 years (Powder)

• Clinical Information:

  No Development Reported

• CAS Number:

  503559-84-0