Products for Research Use Only
RegisterLogin

Metergoline

CAT: 0026-B3088-25Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0026-B3088-25Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Metergoline is a serotonin (5-HT) receptor antagonist. It is active at 5-HT1 (pKi=7.8 for 5-HT1B), 5-HT2 (pKi=8.64, 8.75 and 8.75 for 5-HT2A, 5-HT2B and 5-HT2C respectively) and 5-HT7 (pKi=16 nM) receptor subtypes. Metergoline potently inhibits 5-HT radiolabeling of the human 5-hydroxytryptamine(7) receptor, with an IC₅₀ value of 73 nM. It inhibits 5-HT7 receptor-stimulated cAMP production with an IC₅₀ of 321 nM in HEK293 cells.
Shipping Conditions
RT
Storage Conditions
-20ºC
Shelf Life
36 months

Alternative Products

CatalogName
B6365-100Metergoline
A18261-10Metergoline 10mg
HY-B1033R-01Metergoline (Standard)
A18261-5Metergoline 5mg

Popular Products