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Mepivacaine-d3

CAT: 0804-HY-B0517SSize: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-B0517SSize:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Mepivacaine-d3 is the deuterium labeled Mepivacaine. Mepivacaine is an amide-type local anesthetic agent. Mepivacaine binds to specific voltage-gated sodium ion channels in neuronal cell membranes, which inhibits both sodium influx and membrane depolarization[1][2].
CAS Number
1346597-90-7
UNSPSC
12352005
Target
Sodium Channel
Type
Isotope-Labeled Compounds
Related Pathways
Membrane Transporter/Ion Channel
Field of Research
Neurological Disease
Purity
99.0
Solubility
10 mM in DMSO|DMF : ≥ 30mg/mL|DMSO : ≥ 25mg/mL|Ethanol : ≥ 30mg/mL
Smiles
O=C(C1N(CCCC1)C([2H])([2H])[2H])NC2=C(C=CC=C2C)C
Molecular Formula
C15H19D3N2O
Molecular Weight
249.37
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216. |[2]Froehle M, et al. ECMO for Cardiac Rescue after Accidental Intravenous Mepivacaine Application. Case Rep Pediatr. 2012;2012:491692.|[3]mepivacaine hydrochloride.|[4]Burm, A.G., et al., Pharmacokinetics of the enantiomers of mepivacaine after intravenous administration of the racemate in volunteers. Anesth Analg, 1997. 84 (1) : p. 85-9.|[5]Leffler, A., J. Reckzeh, and C. Nau, Block of sensory neuronal Na+ channels by the secreolytic ambroxol is associated with an interaction with local anesthetic binding sites. Eur J Pharmacol, 2010. 630 (1-3) : p. 19-28.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported

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