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Z8554052021

CAT: 0804-HY-161113Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-161113Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Z8554052021 (compound 2021) is a potent CaSR and indeed GPCR positive allosteric modulator (PAM) with an EC50 of 3.3 nM. Z8554052021 has the potential for hyperparathyroidism research[1].
UNSPSC
12352005
Target
CaSR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/z8554052021.html
Solubility
10 mM in DMSO
Smiles
C[C@H](N[C@@H](C)C1=CC(N2N=CC=C2)=CC=C1)C3=CSC4=C3C=CC=C4
Molecular Formula
C21H21N3S
Molecular Weight
347.48
References & Citations
[1]Fangyu Liu, et al. Structure-based discovery of positive allosteric modulators for the calcium sensing receptor. bioRxiv, December 27, 2023.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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CatalogName
T208983-01Z8554052021

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