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Y08175

CAT: 0804-HY-142743Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-142743Size:1 Each
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Description
Y08175 is a potent CBP bromodomain inhibitor. Y08175 exhibits considerable inhibitory effect with IC50s of 37 and 178.15 nM against CBP bromodomain in AlphaScreen assay and HTRF assay, respectively. Y08175 can be used for the research of prostate cancer[1].
CAS Number
2223014-57-9
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/y08175.html
Solubility
10 mM in DMSO
Smiles
O=C(O)C1=CC(C2=CN(C)N=C2)=C(F)C(NC(C3=CN(C(C)=O)C4=C3C=C(OC)C=C4)=O)=C1
Molecular Formula
C23H19FN4O5
Molecular Weight
450.42
References & Citations
[1]Xiang Q, et al. Design, Synthesis, and Biological Evaluation of 1- (Indolizin-3-yl) ethan-1-ones as CBP Bromodomain Inhibitors for the Treatment of Prostate Cancer. J Med Chem. 2022;65 (1) :785-810.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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CatalogName
T62713-01Y08175

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