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APJ receptor agonist 3

CAT: 0804-HY-139876Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-139876Size:1 Each
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Description
APJ receptor agonist 3 is a potent and orally active APJ receptor agonist with an EC50 value of 0.027 nM.
CAS Number
2759159-56-1
UNSPSC
12352005
Target
Apelin Receptor (APJ)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/apj-receptor-agonist-3.html
Solubility
10 mM in DMSO
Smiles
CCCCC(N(C1=C(C=CC=C1OC)OC)C(O)=C2C(N3C[C@H](C4=CC=C(C=N4)Cl)CC3)=O)=NC2=O
Molecular Formula
C26H29ClN4O5
Molecular Weight
512.99
References & Citations
[1]Pi Z, et al. Identification of 6-Hydroxypyrimidin-4 (1H) -one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists. ACS Med Chem Lett. 2021 Oct 22;12 (11) :1766-1772.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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