PP2A Cancerous-IN-1
CAT:
804-HY-139296
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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PP2A Cancerous-IN-1
- CAS Number: 1403933-79-8
- UNSPSC Description: PP2A Cancerous-IN-1 is a strong and potent CIP2A (Cancerous inhibitor of PP2A) and p-Akt inhibitor. PP2A Cancerous-IN-1 shows the most potent antiproliferative activities[1]. PP2A Cancerous-IN-1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
- Target Antigen: Akt
- Type: Reference compound
- Related Pathways: PI3K/Akt/mTOR
- Applications: Cancer-Kinase/protease
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/pp2a-cancerous-in-1.html
- Solubility: 10 mM in DMSO
- Smiles: C#CC1=CC=CC(NC2=C3C=C(OC)C(OC)=CC3=NC(NC4=CC=C(C=C4)OC5=CC=CC=C5)=N2)=C1
- Molecular Weight: 488.54
- References & Citations: [1]Chen KF, et al. Development of erlotinib derivatives as CIP2A-ablating agents independent of EGFR activity. Bioorg Med Chem. 2012;20(20):6144-6153.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported