Raloxifene 6-Monomethyl Ether
CAT:
804-HY-135584
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

Raloxifene 6-Monomethyl Ether
- CAS Number: 178451-13-3
- UNSPSC Description: Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibits estrogen receptor α. Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with an IC50 of 250 nM and a pIC50 of 6.6[1].
- Target Antigen: Estrogen Receptor/ERR
- Type: Reference compound
- Related Pathways: Vitamin D Related/Nuclear Receptor
- Applications: Metabolism-protein/nucleotide metabolism
- Field of Research: Endocrinology
- Assay Protocol: https://www.medchemexpress.com/raloxifene-6-monomethyl-ether.html
- Solubility: 10 mM in DMSO
- Smiles: O=C(C1=C(C2=CC=C(O)C=C2)SC3=CC(OC)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4
- Molecular Weight: 487.61
- References & Citations: [1]Chang YH, et al. Computational study of estrogen receptor-alpha antagonist with three-dimensional quantitative structure-activity relationship, support vector regression, and linear regression methods. Int J Med Chem. 2013;2013:743139.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported