BRD4 ligand-Linker Conjugate 1

• UNSPSC Description:

  BRD4 ligand-Linker Conjugate 1 is a target protein ligand-linker conjugate that can be used in the synthesis of PROTACs. BRD4 ligand-Linker Conjugate 1 consists of BRD4 Degrader CFT-2718 and

• Target Antigen:

  Target Protein Ligand-Linker Conjugates

• Type:

  Reference compound

• Related Pathways:

  PROTAC

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/brd4-ligand-linker-conjugate-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  ClC1=CC=C(C2=NC3(CC3)C4=NN=C(C)N4C5=CC=C(C6=CN(CCCCCCN)N=C6)C=C25)C=C1

• Molecular Weight:

  500.04

• References & Citations:

  [1]Sun D, et al. Evaluation of the Small-molecule BRD4 Degrader CFT-2718 in Small-cell Lung Cancer and Pancreatic Cancer Models. Mol Cancer Ther. 2021 Aug;20(8):1367-1377.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2154358-89-9