GLP-1 receptor agonist 3

GLP-1 receptor agonist 3

• CAS Number: 2230200-09-4
• UNSPSC Description: GLP-1 receptor agonist 3 (compound (R)-4A-1) is a GLP-1 receptor agonist (WO2018109607A1), used for diabetes research. compound (S)-4A-1 shows EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively[1].
• Target Antigen: GCGR
• Type: Reference compound
• Related Pathways: GPCR/G Protein
• Applications: Metabolism-sugar/lipid metabolism
• Field of Research: Metabolic Disease
• Assay Protocol: https://www.medchemexpress.com/glp-1-receptor-agonist-3.html
• Solubility: 10 mM in DMSO
• Smiles: O=C(C1=CC=C2N=C(CN3CCC(C4=NC(OCC5=CC=C(C#N)C=C5F)=CC=C4)CC3)N(C[C@@H]6OCC6)C2=C1)O
• Molecular Weight: 555.60
• References & Citations: [1]Gary Erik Aspnes, et al. Glp-1 receptor agonists and uses thereof. WO2018109607A1.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported