Eperisone

CAT: 0804-HY-128891Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-128891Size:1 Each
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Description
Eperisone ((±) -Eperisone) is an antispasmodic agent and centrally acting muscle relaxant useful in the study of diseases characterized by muscle stiffness and pain. Eperisone acts by relaxing skeletal and vascular smooth muscle, resulting in vasodilation, decreased muscle tone, improved circulation, and inhibition of pain reflexes. Eperisone is also a potent P2X7 receptor antagonist[1][2][3][4].
CAS Number
[64840-90-0]
UNSPSC
12352005
Target
P2X Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/eperisone.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC=C(CC)C=C1)C(C)CN2CCCCC2
Molecular Formula
C17H25NO
Molecular Weight
259.39
References & Citations
[1]Cabitza P, et al. Efficacy and safety of eperisone in patients with low back pain: a double blind randomized study. Eur Rev Med Pharmacol Sci. 2008 Jul-Aug;12 (4) :229-35.|[2]Frandisco Colomer Rusinvol, et al. Effects of Two Diffferent Doses of Eperisone in the Treatment of Acute Low Back Pain. The Journal of Applied Research.|[3]Bavage S, et al. Clinical efficacy and safety of eperisone for low back pain: A systematic literature review. Pharmacol Rep. 2016 Oct;68 (5) :903-12.|[4]Okada M, et al. Eperisone Hydrochloride, a Muscle Relaxant, Is a Potent P2X7 Receptor Antagonist. Chem Pharm Bull (Tokyo) . 2024;72 (3) :345-348.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Launched

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