Lavoltidine

• Description :

  Lavoltidine (Loxtidine) is an an orally active, irreversible and highly potent histamine H2-receptor antagonist. Lavoltidine strongly inhibits gastric acid secretion and also induces hypergastrinemia[1].

• Product Name Alternative :

  Loxtidine; AH-234844

• UNSPSC :

  12352005

• Target :

  Histamine Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

• Applications :

  Cancer-programmed cell death

• Field of Research :

  Cancer

• Assay Protocol :

  https://www.medchemexpress.com/lavoltidine.html

• Solubility :

  10 mM in DMSO

• Smiles :

  OCC1=NN(C(NCCCOC2=CC=CC(CN3CCCCC3)=C2)=N1)C

• Molecular Formula :

  C19H29N5O2

• Molecular Weight :

  359.47

• References & Citations :

  [1]Takaishi S, et al. Synergistic inhibitory effects of gastrin and histamine receptor antagonists on Helicobacter-induced gastric cancer.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  Phase 1

• Isoform :

  H2 Receptor

• CAS Number :

  [76956-02-0]