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PD125754

CAT: 0804-HY-120756Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-120756Size:1 Each
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Description
PD125754 is an oligopeptide renin inhibitor (IC50: 22 nM) [1].
CAS Number
124339-32-8
UNSPSC
12352005
Target
Renin
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/pd125754.html
Solubility
10 mM in DMSO
Smiles
O=C(OC(C)(C)C)N[C@H]([C@@H](O)CCC(N[C@H]([C@@H](O)CC(N[C@@H](CC(C)C)C(NCC1=CC=CC(CN)=C1)=O)=O)CC2CCCCC2)=O)CC3=CC=CC=C3
Molecular Formula
C42H65N5O7
Molecular Weight
751.99
References & Citations
[1]Cooper J, et al. X-ray crystallographic analysis of inhibition of endothiapepsin by cyclohexyl renin inhibitors. Biochemistry. 1992 Sep 8;31 (35) :8142-50.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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