SR2595

CAT: 0804-HY-116521Size: 5 mgDry Ice: NoHazardous: No

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CAT#:0804-HY-116521Size:5 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Description

SR2595 is an inverse agonist of PPARγ with an IC50 of 30 nM[1].

CAS Number

1415252-61-7

UNSPSC

12352005

Target

PPAR

Type

Reference compound

Related Pathways

Cell Cycle/DNA Damage; Metabolic Enzyme/Protease; Vitamin D Related/Nuclear Receptor

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/sr2595.html

Solubility

10 mM in DMSO

Smiles

CC(N1CC2=CC=C(C=C2)C3=CC=CC=C3C(O)=O)=C(C4=C1C=CC(C(N[C@H](C5=CC=C(C=C5)C(C)(C)C)C)=O)=C4)C

Molecular Formula

C37H38N2O3

Molecular Weight

558.71

References & Citations

[1]Marciano DP, et al. Pharmacological repression of PPARγ promotes osteogenesis. Nat Commun. 2015 Jun 12;6:7443.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

PPARγ

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