Eltenac

• Description:

  Eltenac, a non-steroidal anti-inflammatory drug (NSAID), is a COX inhibitor. Eltenac shows IC50 of 0.03 μM for both COX-1 and COX-2 in isolated human whole blood[1].

• UNSPSC:

  12352005

• Hazard Statement:

  H301

• Target:

  COX

• Type:

  Reference compound

• Related Pathways:

  Immunology/Inflammation

• Applications:

  COVID-19-immunoregulation

• Field of Research:

  Inflammation/Immunology

• Assay Protocol:

  https://www.medchemexpress.com/eltenac.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(O)CC1=CSC=C1NC2=C(Cl)C=CC=C2Cl

• Molecular Formula:

  C12H9Cl2NO2S

• Molecular Weight:

  302.18

• Precautions:

  P264-P270-P330-P405-P501

• References & Citations:

  [1]Klein T, , et al. Characterization of eltenac and novel COX-2 selective thiopheneacetic acid analogues in vitro and in vivo. Biochem Pharmacol. 2008;76 (6) :717-725.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  Phase 1

• Isoform:

  COX-1; COX-2

• CAS Number:

  [72895-88-6]