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Epelsiban

CAT: 0804-HY-105018Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-105018Size:1 Each
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Description
Epelsiban (GSK 557296) is a potent, selective and orally bioavailable oxytocin receptor antagonist, with a pKi of 9.9 for human oxytocin receptor.
CAS Number
872599-83-2
Product Name Alternative
GSK 557296
UNSPSC
12352005
Target
Oxytocin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/GSK_557296.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCOCC1)[C@@H](C2=C(N=C(C)C=C2)C)N3[C@](C(N[C@H](C4CC5=CC=CC=C5C4)C3=O)=O)([H])[C@@H](C)CC
Molecular Formula
C30H38N4O4
Molecular Weight
518.65
References & Citations
[1]Borthwick AD, et al. Pyridyl-2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists: synthesis, pharmacokinetics, and in vivo potency. J Med Chem. 2012 Jan 26;55 (2) :783-96.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 2

Alternative Products

CatalogName
XJB59983-01Epelsiban
A19336-5Epelsiban 5mg
A19336-1Epelsiban 1mg
A19336-50Epelsiban 50mg
A19336-100Epelsiban 100mg
A19336-10Epelsiban 10mg
T31647-01Epelsiban besylate
A19336-25Epelsiban 25mg

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