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Carpindolol

CAT: 0804-HY-103199Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-103199Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Carpindolol (SDZ21009) is a 5-HT1B receptor antagonist (pKd of 8.53 and pKB of 8.0) and a 5-HT1D receptor agonist (pEC50 of 5.91 and pKd of 6.37) [1].
CAS Number
39731-05-0
Product Name Alternative
SDZ21009
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/carpindolol.html
Solubility
10 mM in DMSO
Smiles
O=C(C(N1)=CC2=C1C=CC=C2OCC(O)CNC(C)(C)C)OC(C)C
Molecular Formula
C19H28N2O4
Molecular Weight
348.44
References & Citations
[1]P Schoeffter, et al. 5-Hydroxytryptamine 5-HT1B and 5-HT1D receptors mediating inhibition of adenylate cyclase activity. Pharmacological comparison with special reference to the effects of yohimbine, rauwolscine and some beta-adrenoceptor antagonists. Naunyn Schmiedebergs Arch Pharmacol. 1989 Sep;340 (3) :285-92.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT1 Receptor; mLAG-3

Alternative Products

CatalogName
599099Carpindolol

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