CaMKK2-IN-1

• UNSPSC Description:

  CaMKK2-IN-1 is a selective, ligand-efficient inhibitor of CaMKK2, with IC50 of 7 nM[1].

• Target Antigen:

  Others

• Type:

  Reference compound

• Related Pathways:

  Others

• Applications:

  Cancer-programmed cell death

• Field of Research:

  cancer

• Assay Protocol:

  https://www.medchemexpress.com/camkk2-in-1.html

• Solubility:

  DMSO : 40 mg/mL (ultrasonic;warming;heat to 60°C)

• Smiles:

  CCOC1=CC=C(C(C2=CC(C3CCCC3)=C(C(O)=O)C=C2)=NC=N4)C4=C1

• Molecular Weight:

  362.42

• References & Citations:

  [1]Young Chen, et al. Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2). J Med Chem. 2023 Dec 14;66(23):15750-15760.

• Shipping Conditions:

  Room Temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  3032691-65-6