PIP5K1α-IN-1

• UNSPSC Description:

  PIP5K1α-IN-1 (Compound 3e) is an inhibitor for phosphatidylinositol 4-phosphate 5-kinase type I α (PIP5K1α) with an IC50 of 0.46 μM[1].

• Target Antigen:

  Others

• Type:

  Reference compound

• Related Pathways:

  Others

• Applications:

  Cancer-Kinase/protease

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/pip5k1α-in-1.html

• Solubility:

  10 mM in DMSO

• Smiles:

  CC(C1=C(C=CC2=C1CC[C@@]3([H])C(C)(CCC[C@]23C)C)OCC4=CN(N=N4)C5=CC([N+]([O-])=O)=CC=C5)C

• Molecular Weight:

  488.62

• References & Citations:

  [1]Haidar S, et al. “1,2,3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors.” Bioorganic & medicinal chemistry vol. 105 (2024): 117727.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  3063813-76-0