GDC 0941
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No








GDC 0941
Background:
GDC 0941 is a potent inhibitor of the PI 3-kinase family. Specifically, GDC 0941 has been shown to inhibit PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ.Description:
Pan-PI3K kinase inhibitorProduct Name Alternative:
Pictrelisib, Pictilisib, GNE 0941, 2-​ (1H-​indazol-​4-​yl) -​6-​[[4-​ (methylsulfonyl) -​1-​piperazinyl]methyl]-​4-​ (4-​morpholinyl) -​thieno[3, ​2-​d]pyrimidineUNSPSC:
41116105Type:
InhibitorSource:
SyntheticField of Research:
Cell Signaling | Cancer | Apoptosis | Cancer Growth Inhibitors | Tyrosine Kinase InhibitorsPurity:
≥98%Weight:
0.025Format:
White solidSolubility:
Soluble in DMSOMolecular Formula:
C23H27N7O3S2Molecular Weight:
513.63Precautions:
Not for use in humans. Not for use in diagnostics or therapeutics. For in vitro research use only.References & Citations:
1. Zheng J., Wang H., Yao J., & Zou X. (2014) Die Pharmazie. 69(1): 38–42.CAS Number:
957054-30-7
