Products for Research Use Only
RegisterLogin

Gallopamil

CAT: 0804-HY-14276-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-14276-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Gallopamil (Methoxyverapamil), a methoxy derivative of Verapamil, is a phenylalkylamine calcium antagonist[1]. Gallopamil inhibits acid secretion in a concentration-dependent manner with an IC50 of 10.9 μM[2]. Gallopamil is a potent antiarrhythmic and vasodilator agent[3].
CAS Number
16662-47-8
Product Name Alternative
Methoxyverapamil
UNSPSC
12352005
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/gallopamil.html
Purity
98.0
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
COC1=C(OC)C(OC)=CC(C(CCCN(C)CCC2=CC(OC)=C(OC)C=C2)(C#N)C(C)C)=C1
Molecular Formula
C28H40N2O5
Molecular Weight
484.63
References & Citations
[1]Brogden RN, et al. Gallopamil. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in ischaemic heart disease. Drugs. 1994 Jan;47 (1) :93-115.|[2]Sewing KF, et al. Calcium channel antagonists verapamil and gallopamil are powerful inhibitors of acid secretion in isolated and enriched guinea pig parietal cells. Pharmacology. 1983;27 (1) :9-14.|[3]Kirchengast M, et al. Reperfusion arrhythmias in closed-chest rats: the effect of myocardial noradrenaline depletion and Ca2 (+) -antagonism. Clin Exp Pharmacol Physiol. 1991 Apr;18 (4) :217-21.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
Calcium Channel

Alternative Products

CatalogName
MBS3614868-01Gallopamil
GTR19200287-01Gallopamil, (-) -
MBS5773837Gallopamil, (-)-
A21229-25Gallopamil 25mg
A21229-1Gallopamil 1mg
GTR19177331-01Gallopamil hydrochloride
A21229-500Gallopamil 500mg
A21229-10Gallopamil 10mg
GTR19200288-01Gallopamil HCl, (-) -
A21229-100Gallopamil 100mg

Popular Products