Cyamemazine

CAT: 0804-HY-14264-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-14264-01Size:5 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
Cyamemazine is a neuroleptic agent that contains the phenothiazine chromophore. Cyamemazine is often used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki of 12 nM), 5-HT2A (Ki = 1.5 nM) and 5-HT2C (Ki of 75 nM) receptors antagonist with antipsychotic activity[1][2].
CAS Number
[3546-03-0]
UNSPSC
12352005
Hazard Statement
H410
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cyamemazine.html
Purity
99.42
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
CN(C)CC(C)CN1C2=C(C=CC(C#N)=C2)SC3=CC=CC=C31
Molecular Formula
C19H21N3S
Molecular Weight
323.46
Precautions
H410
References & Citations
[1]Bourin M, et al. Preclinical and clinical pharmacology of cyamemazine: anxiolytic effects and prevention of alcohol and benzodiazepine withdrawal syndrome. CNS Drug Rev. 2004 Fall;10 (3) :219-29.|[2] Vendrell-Criado V, et al. Photobehavior of the antipsychotic drug cyamemazine in a supramolecular gel protective environment. J Photochem Photobiol B. 2020 Jan;202:111686.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor; lactoferrin; α-1 microglobulin

Alternative Products

CatalogName
BA5030-10Cyamemazine
TRC-C951502-1MGCyamemazine-d6
TRC-C951570-25MGCyamemazine Sulfoxide
RM-C250150-01Cyamemazine Maleate
RM-C250151-01Cyamemazine Tartrate
RM-C250101-01Cyamemazine Cyano Impurity
RM-C250152-01Cyamemazine Impurity 2
RM-C250153-01Cyamemazine Impurity 3
TRC-N754860-100MGN-Nitroso Cyamemazine Impurity

Popular Products