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AP102

CAT: 0804-HY-P2434Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-P2434Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA) . AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC50: 0.63 and 0.65 nM, respectively) . AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research[1].
CAS Number
846569-60-6
UNSPSC
12352209
Target
Somatostatin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Cancer; Metabolic Disease; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ap102.html
Solubility
H2O
Smiles
O=C(N[C@H](C(N[C@H](C(N1)=O)C(C)C)=O)CCCCN)[C@H](NC([C@@H](NC([C@H](CSSC[C@H]1C(N[C@H](C(N)=O)[C@H](O)C)=O)NC([C@H](N)CC(C=C2)=CC(I)=C2N)=O)=O)CC(C=C3)=CC(I)=C3O)=O)CC4=CNC5=CC=CC=C45
Molecular Formula
C50H66I2N12O10S2
Molecular Weight
1313.07
References & Citations
[1]Tarasco E, et al. Effect of AP102, a subtype 2 and 5 specific somatostatin analog, on glucose metabolism in rats. Endocrine. 2017 Oct;58 (1) :124-133.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
SSTR2; SSTR5

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