Apatinib

• Description:

  VEGFR2 inhibitor, orally bioavailable, selective

• Product Name Alternative:

  N-[4-(1-cyanocyclopentyl)phenyl]-2-(pyridin-4-ylmethylamino)pyridine-3-carboxamide;methanesulfonic acid

• Field of Research:

  Tyrosine Kinase VEGFR

• Purity:

  0.9985

• Form:

  A solid

• Solubility:

  ≥49.4 mg/mL in DMSO; insoluble in H2O; ≥2.17 mg/mL in EtOH with gentle warming and ultrasonic

• Smiles:

  CS(=O)(=O)O.C1CCC(C1)(C#N)C2=CC=C(C=C2)NC(=O)C3=C(N=CC=C3)NCC4=CC=NC=C4

• Molecular Formula:

  C25H27N5O4S

• Molecular Weight:

  493.58

• Shipping Conditions:

  Blue ice

• Storage Conditions:

  Store at -20°C.

• CAS Number:

  1218779-75-9