EPZ-6438

• Description:

  EZH2 inhibitor, potent and selective

• Product Name Alternative:

  N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-5-[4-(morpholin-4-ylmethyl)phenyl]benzamide

• Sequence:

  E-7438

• Field of Research:

  Chromatin Epigenetics Histone Methyltransferase

• Purity:

  0.9942

• Form:

  A solid

• Solubility:

  ≥28.64 mg/mL in DMSO; insoluble in EtOH; insoluble in H2O

• Smiles:

  CCN(C1CCOCC1)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C4=CC=C(C=C4)CN5CCOCC5

• Molecular Formula:

  C34H44N4O4

• Molecular Weight:

  572.74

• Shipping Conditions:

  Blue ice

• Storage Conditions:

  Desiccate at -20°C.

• CAS Number:

  1403254-99-8